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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'BDKRB2' and Ligand = 'BDBM50067261'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
BDKRB2


(Homo sapiens (Human))
BDBM50067261
PNG
(CHEMBL556816 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...)
Show SMILES CN(C(=O)CNC(=O)Nc1cccc(Cl)c1)c1ccc(Cl)c(COc2cccn3c(Br)c(C)nc23)c1Cl
Show InChI InChI=1S/C25H21BrCl3N5O3/c1-14-23(26)34-10-4-7-20(24(34)31-14)37-13-17-18(28)8-9-19(22(17)29)33(2)21(35)12-30-25(36)32-16-6-3-5-15(27)11-16/h3-11H,12-13H2,1-2H3,(H2,30,32,36)
UniProtKB/SwissProt

antibodypedia
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 3.80n/an/an/an/an/an/a



Fujisawa Pharmaceutical Company, Ltd

Curated by ChEMBL


Assay Description
Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.


J Med Chem 41: 4053-61 (1998)


Article DOI: 10.1021/jm980214f
BindingDB Entry DOI: 10.7270/Q2WQ04GV
More data for this
Ligand-Target Pair