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Found 2 Enz. Inhib. hit(s) with Target = 'Bcl-2-like protein 1' and Ligand = 'BDBM174843'
TargetBcl-2-like protein 1(Homo sapiens (Human))
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174843(US9115061, VIII)
Affinity DataIC50:  160nMT: 2°CAssay Description:A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes) and purified ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBcl-2-like protein 1(Homo sapiens (Human))
Burnham Institute For Medical Research

US Patent
LigandPNGBDBM174843(US9115061, VIII)
Affinity DataKd:  2.75E+3nMpH: 7.4Assay Description:Titrations were performed using a VP-ITC or ITC200 calorimeter from Microcal (Northampton, Mass.). BCL-XL was used at concentrations between 25 and 1...More data for this Ligand-Target Pair
In DepthDetails US Patent