Found 33 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM25392' 
Affinity DataKi: 80nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataKi: 670nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]-dihydroalprenolol from beta-1 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataKi: 1.59E+3nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Compound was evaluated in vitro for beta-adrenergic activity against beta-1 adrenergic receptor by the inhibition of insulin stimulated [14C]- glucos...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Compound was evaluated for its binding affinity towards beta-1 adrenergic receptor in rat heart membrane by displacing [125I]- iodocyanopindololMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at beta1 adrenoceptor (unknown origin) expressed in HEK293 cells assessed as cAMP accumulation incubated for 60 mins by microplate r...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human adrenergic beta1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human beta1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.0840nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 12nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as increase in cAMP production after 2 days by radioimmun...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoass...Checked by AuthorMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 12nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoass...Checked by AuthorMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation afte...More data for this Ligand-Target Pair
Affinity DataEC50: 980nMAssay Description:Effective concentration against 125I]iodocyanopindolol(ICYP) binding to beta adrenergic receptor was determinedMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at recombinant human beta1 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human beta1 adrenergic receptor expressed in HEK293 cells assessed as increase in cAMP accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human beta1 adrenergic receptor expressed in HEK293 cells assessed as increase in cAMP accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human beta1 adrenoreceptor overexpressed in human HEK293 cells assessed as cAMP accumulation incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human beta1 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 100nMAssay Description:Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.0840nMAssay Description:Agonist activity at human cloned adrenergic beta1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.0840nMAssay Description:Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1nMAssay Description:Activity against human beta 1 adrenergic receptor (AR), expressed in CHO cells.More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.0840nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 1nMAssay Description:Activity at human beta-1 adrenergic receptor expressed in CHO cells by stimulation of cAMP productionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonistic activity (beta-1 adrenergic receptor) for the percent maximal increase in contraction rate of isolated guinea pig atriaMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
UniversitÄT WÜRzburg
Curated by PDSP Ki Database
Affinity DataEC50: 0.0840nMAssay Description:Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
