Affinity DataKi: 34nMAssay Description:Binding inhibition constant was determined by inhibition of [125I]-iodocyanopindolol binding to Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Agonistic activity was determined by measuring cAMP accumulation in CHO cells expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair