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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50296957'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296957(4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan...)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human adrenergic beta3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50296957(4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at dog recombinant adrenergic beta3 receptor expressed in CHO cells assessed as stimulation of cAMP level after 1 hr by enzyme immun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Heptares Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296957(4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan...)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human recombinant adrenergic beta3 receptor expressed in CHO cells assessed as stimulation of cAMP level after 1 hr by enzyme imm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed