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Found 1 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50296959'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50296959(3-(cyclohexyloxy)-4'-((S)-3-hydroxy-2-((R)-2-hydro...)
Affinity DataEC50:  0.820nMAssay Description:Agonist activity at human recombinant adrenergic beta3 receptor expressed in CHO cells assessed as stimulation of cAMP level after 1 hr by enzyme imm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed