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Found 4 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 5' and Ligand = 'BDBM50124940'
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50124940((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4'-methyl-[1,4'...)
Affinity DataKi:  47.6nMAssay Description:Inhibitory activity against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50124940((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4'-methyl-[1,4'...)
Affinity DataKi:  93nMAssay Description:Inhibitory activity of the compound against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50124940((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4'-methyl-[1,4'...)
Affinity DataKi:  97.8nMAssay Description:Inhibitory activity of the compound against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50124940((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4'-methyl-[1,4'...)
Affinity DataKi:  98nMAssay Description:Inhibitory activity against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed