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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50078762'
TargetCannabinoid receptor 2(MOUSE)
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Hawaii At Manoa

Curated by ChEMBL
LigandPNGBDBM50078762(CHEMBL3416121)
Affinity DataEC50:  16nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed