Found 3 Enz. Inhib. hit(s) with Target = 'Carnitine O-palmitoyltransferase 1, liver isoform' and Ligand = 'BDBM61402'
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of CPT1 in rat cardiac mitochondria using [3H]carnitine by radiometric methodMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 1.48E+5nMAssay Description:Inhibition of CPT1 in rat liver mitochondria using [3H]carnitine by radiometric methodMore data for this Ligand-Target Pair