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Found 1 Enz. Inhib. hit(s) with Target = 'Class D beta-lactamase' and Ligand = 'BDBM50021954'
TargetClass D beta-lactamase(Brachyspira pilosicoli)
Institut Pasteur

Curated by ChEMBL
LigandPNGBDBM50021954((2S,5R)-3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Brachyspira pilosicoli beta-lactamase OXA-63 expressed in Escherichia coli BL21 (DE3) assessed as reduction in nitrocefin hydrolysis by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed