Affinity DataKi: 0.660nM ΔG°: -51.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound (isomer) was tested in the absence of light for inhibitory activity against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound was tested for inhibitory activity against human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:In vitro inhibition of human coagulation factor Xa (Xa) in a purified enzyme system.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity of the compound was evaluated against Coagulation factor XMore data for this Ligand-Target Pair