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Found 3 Enz. Inhib. hit(s) with Target = 'Cystic fibrosis transmembrane conductance regulator' and Ligand = 'BDBM50244767'
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50244767(4-((4-oxo-2-thioxo-3-(3-(trifluoromethyl)phenyl)th...)
Affinity DataIC50:  300nMAssay Description:Inhibition of CFTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50244767(4-((4-oxo-2-thioxo-3-(3-(trifluoromethyl)phenyl)th...)
Affinity DataIC50:  300nMAssay Description:Inhibition of CFTRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50244767(4-((4-oxo-2-thioxo-3-(3-(trifluoromethyl)phenyl)th...)
Affinity DataIC50:  380nMAssay Description:Inhibition of human wild type CFTR expressed in rat FRT cells assessed as chloride current by short-circuit current measurementsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed