Affinity DataKi: 2.40nMAssay Description:Inhibition of [3H]SCH-23,390 binding to Dopamine receptor D1 at 0.25 nMMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 from canine striatumMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Antagonist activity at recombinant human D1 receptor expressed in CHOK1 cells assessed as inhibition of SKF81297-induced beta arrestin2 recruitment p...More data for this Ligand-Target Pair