TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences
Curated by ChEMBL
National Institute Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Binding affinity against Opioid receptor delta 1 in P2 membrane preparation of rat brain by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences
Curated by ChEMBL
National Institute Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Compound was tested for its binding affinity against opioid receptor delta using [3H]-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences
Curated by ChEMBL
National Institute Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 2.13nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences
Curated by ChEMBL
National Institute Of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Inhibition of [3H]- ]DSLET binding to delta receptor from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.695nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 98.3nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair