Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataEC50: 0.620nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey methodMore data for this Ligand-Target Pair
Affinity DataEC50: 0.410nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair