Affinity DataKi: 99nMAssay Description:Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cell membrane incubated for 1 hr by TopCount scintillation cou...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Agonist activity at delta opioid receptor in Swiss Webster albino mouse vas deferans assessed as inhibition of electrically-induced longitudinal musc...More data for this Ligand-Target Pair