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Found 3 Enz. Inhib. hit(s) with Target = 'Deoxyribonuclease gamma' and Ligand = 'BDBM50206432'
TargetDeoxyribonuclease gamma(Homo sapiens (Human))
University Of Nis

Curated by ChEMBL
LigandPNGBDBM50206432(4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of DNase gamma (unknown origin) transfected in HeLa S3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyribonuclease gamma(Homo sapiens (Human))
University Of Nis

Curated by ChEMBL
LigandPNGBDBM50206432(4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human recombinant DNase gamma expressed in Rosetta DE3 cells assessed as increase in acidsoluble DNA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxyribonuclease gamma(Homo sapiens (Human))
University Of Nis

Curated by ChEMBL
LigandPNGBDBM50206432(4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of DNase gamma-mediated HMGB1 release expressed in human staurosporine-induced HeLaS3 cells treated 1 hr before staurosporine challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed