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Found 4 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM50324514'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324514((+)-Ethyl 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324514((+)-Ethyl 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324514((+)-Ethyl 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7...)
Affinity DataKi:  11.7nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324514((+)-Ethyl 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7...)
Affinity DataIC50:  0.700nMAssay Description:The HypoGen module in DS2.5 was employed to produce pharmaphores with the training set compounds.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed