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Found 2 Enz. Inhib. hit(s) with Target = 'Ecdysone receptor' and Ligand = 'BDBM50326776'
TargetEcdysone receptor(Drosophila melanogaster)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  1.29nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
TargetEcdysone receptor(Lucilia cuprina)
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | CHEM...)
Affinity DataIC50:  900nMAssay Description:Binding affinity to Lucilia cuprina recombinant ecdysone receptor ligand binding domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair