Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50157483'
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157483(4-(1-cyclopentyl-7-fluoro-1H-indazol-3-yl)phenol |...)
Affinity DataIC50:  18nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NFkappaB transcriptionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157483(4-(1-cyclopentyl-7-fluoro-1H-indazol-3-yl)phenol |...)
Affinity DataEC50:  330nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed