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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 2' and Ligand = 'BDBM50426293'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Excitatory amino acid transporter 2


(Homo sapiens (Human))
BDBM50426293
PNG
(CHEMBL2312400)
Show SMILES N[C@@H](C[C@@H](CCC(=O)N1CCCCC1)C(O)=O)C(O)=O
Show InChI InChI=1/C13H22N2O5/c14-10(13(19)20)8-9(12(17)18)4-5-11(16)15-6-2-1-3-7-15/h9-10H,1-8,14H2,(H,17,18)(H,19,20)/t9-,10+/s2
UniProtKB/SwissProt

GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a>3.00E+5n/an/an/an/an/an/a



University of Copenhagen

Curated by ChEMBL


Assay Description
Inhibition of human EAAT2 expressed in HEK293 cells by [3H]-D-Asp uptake assay


J Med Chem 56: 1614-28 (2013)


Article DOI: 10.1021/jm301433m
BindingDB Entry DOI: 10.7270/Q23F4R0N
More data for this
Ligand-Target Pair