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Found 2 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 3' and Ligand = 'BDBM50102486'
TargetExcitatory amino acid transporter 3(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102486(2-Phenyl-4,5-dihydro-oxazole-4,5-dicarboxylic acid...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in absence of L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50102486(2-Phenyl-4,5-dihydro-oxazole-4,5-dicarboxylic acid...)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibitory activity against EAAC1 (EAAT3) in presence of 20 uM L-glutamic acid in mammalian cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed