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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 3' and Ligand = 'BDBM50173935'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Excitatory amino acid transporter 3


(Homo sapiens (Human))
BDBM50173935
PNG
(2-Amino-N-biphenyl-4-yl-succinamic acid | CHEMBL19...)
Show SMILES NC(CC(=O)Nc1ccc(cc1)-c1ccccc1)C(O)=O
Show InChI InChI=1/C16H16N2O3/c17-14(16(20)21)10-15(19)18-13-8-6-12(7-9-13)11-4-2-1-3-5-11/h1-9,14H,10,17H2,(H,18,19)(H,20,21)
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KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 1.00E+3n/an/an/an/an/an/a



Wyeth Research

Curated by ChEMBL


Assay Description
Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 3


Bioorg Med Chem Lett 15: 4985-8 (2005)


Article DOI: 10.1016/j.bmcl.2005.08.003
BindingDB Entry DOI: 10.7270/Q25H7FSP
More data for this
Ligand-Target Pair