Found 5 Enz. Inhib. hit(s) with Target = 'G-protein coupled estrogen receptor 1' and Ligand = 'BDBM17292' TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of E2-Alexa633 from GFP-tagged GPR30 expressed in COS7 cells by FACSMore data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Inhibition of estrogen binding to GPR30 (unknown origin)More data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive binding of estrogen to GPR30 and ER alpha were conducted using COS-7 cells transfected with GPR30-GFP or ER alpha-GFP and fluorescent est...More data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at GPR30 (unknown origin) by calcium mobilization assayMore data for this Ligand-Target Pair
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
University Of New Mexico Health Sciences Center
Curated by ChEMBL
University Of New Mexico Health Sciences Center
Curated by ChEMBL
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at GFP-tagged GPR30 expressed in COS7 cells assessed as half life for increase in intracellular calcium level by spectrofluorimetryMore data for this Ligand-Target Pair
