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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'G-protein coupled receptor 119 (GPR119)' and Ligand = 'BDBM50387908'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G-protein coupled receptor 119 (GPR119)


(Homo sapiens (Human))
BDBM50387908
PNG
(CHEMBL2058669)
Show SMILES CC(C)c1noc(n1)N1CCC(CCCNc2ccc3c(O)coc3c2)CC1
Show InChI InChI=1S/C21H28N4O3/c1-14(2)20-23-21(28-24-20)25-10-7-15(8-11-25)4-3-9-22-16-5-6-17-18(26)13-27-19(17)12-16/h5-6,12-15,22,26H,3-4,7-11H2,1-2H3
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a 73n/an/an/an/a



Sanwa Kagaku Kenkyusho Co., Ltd

Curated by ChEMBL


Assay Description
Agonist activity at human GPR119 receptor expressed in CHO-K1 cells assessed as cAMP accumulation after 30 mins by HTRF assay


Bioorg Med Chem Lett 22: 5123-8 (2012)


Article DOI: 10.1016/j.bmcl.2012.05.117
BindingDB Entry DOI: 10.7270/Q2TD9ZC4
More data for this
Ligand-Target Pair