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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM50346059'
TargetHistamine H1 receptor(Homo sapiens (Human))
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50346059(2,8-dimethyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tet...)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human histamine H1 receptor in SK-N-SH cells assessed as inhibition of histamine-induced calcium level increase during phase-1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50346059(2,8-dimethyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tet...)
Affinity DataIC50:  3.98E+3nMAssay Description:Antagonist activity at human histamine H1 receptor in SK-N-SH cells assessed as inhibition of histamine-induced calcium flow during phase-II compound...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed