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Found 4 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM86741'
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86741(UR-AK59)
Affinity DataKd:  2.34E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea pig ileum assessed as inhibition of histamine-induced positive chronotropic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed