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Found 6 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50127607'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity was measured against Histamine H3 receptor on rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataKi:  42nMAssay Description:Affinity against rat Histamine H3 receptor using [3H]-N-alpha-methyl histamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataKi:  68nMAssay Description:Inhibitory activity measured by [3H]- N alpha- methyl-histamine binding to membranes of SK-N-MC cells expressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataEC50:  724nMAssay Description:Inhibition of human Histamine H3 receptor using [3H]-N-alpha-methyl histamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127607((1R,2R)-2-(1H-Imidazol-4-yl)-cyclopropylamine | (1...)
Affinity DataEC50:  58nMAssay Description:Inhibitory activity determined by the inhibition of cAMP- stimulated beta-galactosidase transcription in SK-N-MC cells expressing the human Histamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed