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Found 2 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 1' and Ligand = 'BDBM178098'
TargetHistone deacetylase 1(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM178098(BRD4097 | US11377423, Compound 9)
Affinity DataIC50: >3.30E+4nMAssay Description:The following non-trypsin coupled in-vitro HDAC enzymatic endpoint assay was used to assay the compounds of the invention. Below is a standardized pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
The Broad Institute

US Patent
LigandPNGBDBM178098(BRD4097 | US11377423, Compound 9)
Affinity DataIC50: >3.33E+4nMpH: 7.4 T: 2°CAssay Description:Purified HDAC1-9 (0.5~5 nM) were incubated with 2 μM carboxyfluorescein (FAM)-labeled acetylated peptide substrate A or B and test compound for ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed