Found 7 Enz. Inhib. hit(s) with Target = 'Insulin receptor' and Ligand = 'BDBM482158' 
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human InsR using myelin basic protein as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of TEL-fused insulin receptor (unknown origin) expressed in mouse BAF3 cells after 2 to 3 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetInsulin receptor(Rattus norvegicus (rat))
Genomics Institute Of The Novartis Research Foundation
Curated by ChEMBL
Genomics Institute Of The Novartis Research Foundation
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of InsR phosphorylation in rat H4-2E cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant InsRMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Inhibition of InsR by cellular assayMore data for this Ligand-Target Pair
