TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Opioid receptor kappa 1 was determined using U69,593 as the radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Clinical Research Institute of Montreal
Curated by PDSP Ki Database
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Opioid receptor kappa 1 of guinea pig brain membranes using 1 nM of (-)-[3H]ethylketazocine as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 80nMAssay Description:Activation of kappa opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 80nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 80nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for...More data for this Ligand-Target Pair