Found 5 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50130757' TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]-U-69593 from kappa opioid receptor in guinea pig brain membrane after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]U-69,593 from KOR in guinea pig brain membranes after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Agonist activity at kappa opioid receptor in human HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
