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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50335568'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335568((1-{4-[2-(3-Methylpiperazin-1-yl)-1H-benzimidazol-...)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]enadoline from human KOP receptor expressed in HEK-293 cells after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335568((1-{4-[2-(3-Methylpiperazin-1-yl)-1H-benzimidazol-...)
Affinity DataEC50:  366nMAssay Description:Agonist activity at human KOP receptor expressed in HEK-293 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed