Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50335569'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335569(1-{1-[1-(Hydroxymethyl)cyclooctyl]piperidin-4-yl}-...)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]enadoline from human KOP receptor expressed in HEK-293 cells after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50335569(1-{1-[1-(Hydroxymethyl)cyclooctyl]piperidin-4-yl}-...)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human KOP receptor expressed in HEK-293 cells assessed as induction of [35S]GTPgammaS binding after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed