Affinity DataKi: 2nMAssay Description:Affinity at K opioid receptor on membranes prepared from guinea pig cerebellum by [3H]- 69593 displacement.More data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Agonist activity at human kappa opioid receptor expressed in COS7 cells after 60 mins IP1 assayMore data for this Ligand-Target Pair