Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50374638'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Mclean Hospital

Curated by ChEMBL
LigandPNGBDBM50374638(CHEMBL258285)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Mclean Hospital

Curated by ChEMBL
LigandPNGBDBM50374638(CHEMBL258285)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed