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Found 6 Enz. Inhib. hit(s) with Target = 'Mas-related G-protein coupled receptor member X1' and Ligand = 'BDBM50497459'
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Mus musculus)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed