BindingDB PrimarySearch_ki

Found 16 Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM17055'

Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Ki: 9.20E+5nM ΔG°: -17.3kJ/molepH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 4.10E+3nMAssay Description:Binding constant for KIT(A829P) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 1.50E+3nMAssay Description:Binding constant for KIT(D816H) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 760nMAssay Description:Binding constant for KIT(D816V) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 7.90E+3nMAssay Description:Binding constant for KIT(L576P) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT(V559D,V654A) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT(V559D) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT(V559D,V654A) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 920nMAssay Description:Binding constant for KIT(D816V) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 380nMAssay Description:Average Binding Constant for KIT; NA=Not Active at 10 uMMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT(V559D) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding constant for KIT(V559D,T670I) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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Details Article PubMed

Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: >1.00E+4nMAssay Description:Binding affinity to human KIT incubated for 1 hr by kinase binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway
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Mast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay

PNG

BDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)

Kd: 9.80E+3nMAssay Description:Binding constant for KIT(V559D,T670I) kinase domainMore data for this Ligand-Target Pair

PDB Reactome pathway
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