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Found 4 Enz. Inhib. hit(s) with Target = 'Menin' and Ligand = 'BDBM152211'
TargetMenin(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50:  1.20E+3nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMenin(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of FITC-MBM1 from menin (unknown origin) measured after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMenin(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50:  1.90E+3nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMenin(Homo sapiens (Human))
University Of Michigan

US Patent
LigandPNGBDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50:  1.90E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In DepthDetails US Patent