Found 8 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50030630'
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataKi: 2.14E+5nMAssay Description:Agonist potency against cloned human metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataIC50: 7.00E+3nMAssay Description:Ability to inhibit mGluR1-alpha-mediated PI (phospho inosotol) hydrolysis was determined at BHK cells at 100 Micro M ConcentrationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataIC50: 2.14E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataIC50: 2.14E+5nMAssay Description:Inhibitory concentration of the compound for half maximal inhibition of PI hydrolysis (mGluR1a)More data for this Ligand-Target Pair