Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50177054'
TargetMetabotropic glutamate receptor 1(RAT)
Biocampus

Curated by ChEMBL
LigandPNGBDBM50177054(9-(1'-cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-th...)
Affinity DataIC50:  43nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50177054(9-(1'-cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-th...)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at human mGluR1 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed