Found 4 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50151897'
Affinity DataKi: >600nMAssay Description:Displacement of [3H]-3-methoxy-5-(pyridin-2-ylethynyl)pyridine from glutamate 5 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >600nMAssay Description:Ability to displace [3H]-3-methoxy-5-(pyridin-2-ylethynyl)pyridine from binding to metabotropic glutamate receptor 5 in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:In vitro functional activity measured by changes in cytosolic [Ca2+] concentrations against rat metabotropic glutamate receptor 5More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory concentration towards human glutamate receptor 5 in calcium flux assayMore data for this Ligand-Target Pair