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Found 3 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50156082'
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Merck

Curated by ChEMBL
LigandPNGBDBM50156082(CHEMBL362969 | N-(4-bromo-2-((1,3-dioxoisoindolin-...)
Affinity DataEC50: <1.00E+3nMAssay Description:Activity at rat mGluR5 expressed in CHO cells assessed as potentiation of glutamate response by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50156082(CHEMBL362969 | N-(4-bromo-2-((1,3-dioxoisoindolin-...)
Affinity DataEC50:  750nMAssay Description:Activity at human mGluR5 expressed in CHO cells assessed as potentiation of glutamate response by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50156082(CHEMBL362969 | N-(4-bromo-2-((1,3-dioxoisoindolin-...)
Affinity DataEC50:  740nMAssay Description:Effective concentration against metabotropic glutamate receptor 5 of human transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed