TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.00240nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.403nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in HEK293 cells incubated for 120 mins by radiometric scintillation ana...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in HEK293 cell membranes incubated for 60 minsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [125I]-IBNalA from MOR-1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DAMGO from human recombinant Opioid receptor mu 1 on CHO cell membranes.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Binding affinity for mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]DAMGO from MOR in HEK293 cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Displacement of [3H]-Diprenorphine from human mu opiod receptor expressed in CHO cells incubated for 1 hr by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Binding affinity against Opioid receptor mu 1 in P2 membrane preparation of rat brain by [3H]DAGO displacement.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]DAMGO from mouse whole brain MORMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.850nMAssay Description:Displacement of [3H]DPDPE from rat mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Displacement of [3H]DAMGO from Sprague-Dawley rat mu opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor expressed in HEK293 cells by visible spectrophotometryMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of radiolabeled DAMGO from mu opioid receptor in Hartley guinea pig brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes incubated for 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity against Opioid receptor mu 1 by displacement of radioligand [3H]-DAGO in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant opioid mu receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting anal...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK293 cells preincubated for 1 hr followed by radioligand addition measured after 1 hr by liqu...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cell membranes after 2 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity to MOR (unknown origin) assessed as inhibition constant by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-DAMGO from Sprague-Dawley rat brain membrane mu opioid receptor incubated for 45 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK293 cell membranes incubated for 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK293 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Illinois At Chicago
Curated by ChEMBL
University Of Illinois At Chicago
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]-IBOxyA from MOR-1 expressed in CHO cellsMore data for this Ligand-Target Pair