Affinity DataKi: 0.190nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]-DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of [3H]-DAMGO to opioid receptor mu of rat fore brain membranes was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.88nMAssay Description:Binding affinity towards Opioid receptor mu 1 expressed in CHO cells was determined by using[3H]DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Opioid receptor mu 1 in guinea pig brain homogenate using [3H]- PL-17 as radioligandMore data for this Ligand-Target Pair