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Found 5 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50108918'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliary

Curated by ChEMBL
LigandPNGBDBM50108918((2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethyl...)
Affinity DataKi:  47nMAssay Description:Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliary

Curated by ChEMBL
LigandPNGBDBM50108918((2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethyl...)
Affinity DataKi:  47.1nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliary

Curated by ChEMBL
LigandPNGBDBM50108918((2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethyl...)
Affinity DataKi:  47.5nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50108918((2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethyl...)
Affinity DataIC50:  4.74E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50108918((2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed