Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50183552'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183552(CHEMBL412331 | H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-...)
Affinity DataKi:  0.920nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183552(CHEMBL412331 | H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-...)
Affinity DataIC50:  200nMAssay Description:Agonist activity at mu opioid receptor by inhibition of muscle contraction in electrically stimulated isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183552(CHEMBL412331 | H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-...)
Affinity DataEC50:  14nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50183552(CHEMBL412331 | H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-...)
Affinity DataEC50:  14nMAssay Description:Inhibition of [35S]GTP-gamma-S binding to rat mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed