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Compile Data Set for Download or QSAR

Found 2 hits Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor' and Ligand = 'BDBM50229584'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Muscarinic acetylcholine receptor


(RAT)
BDBM50229584
PNG
(PILOCARBINE)
Show SMILES CC[C@H]1[C@H](COC1=O)c1cncn1C
Show InChI InChI=1S/C10H14N2O2/c1-3-7-8(5-14-10(7)13)9-4-11-6-12(9)2/h4,6-8H,3,5H2,1-2H3/t7-,8-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
83n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]- Oxo-M binding to muscarinic acetylcholine receptor of rat brain membrane preparations


J Med Chem 35: 2184-91 (1992)


Article DOI: 10.1021/jm00090a006
BindingDB Entry DOI: 10.7270/Q2B27T74
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor


(RAT)
BDBM50229584
PNG
(PILOCARBINE)
Show SMILES CC[C@H]1[C@H](COC1=O)c1cncn1C
Show InChI InChI=1S/C10H14N2O2/c1-3-7-8(5-14-10(7)13)9-4-11-6-12(9)2/h4,6-8H,3,5H2,1-2H3/t7-,8-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
1.01E+3n/an/an/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]QNB binding to muscarinic acetylcholine receptor of rat heart membrane preparation.


J Med Chem 35: 2184-91 (1992)


Article DOI: 10.1021/jm00090a006
BindingDB Entry DOI: 10.7270/Q2B27T74
More data for this
Ligand-Target Pair