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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50008071'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50008071(5-methylfurmethide | CHEMBL92387 | Trimethyl-(5-me...)
Affinity DataIC50:  1.41E+3nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed