Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50323691'
TargetMuscarinic acetylcholine receptor M4(RAT)
Dvanderbilt Program In Drug Discovery
Curated by ChEMBL
Dvanderbilt Program In Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 10 uM acetylcholine-induced calciu...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Dvanderbilt Program In Drug Discovery
Curated by ChEMBL
Dvanderbilt Program In Drug Discovery
Curated by ChEMBL
Affinity DataEC50: 0.000339nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair